Peptide · Research Monograph · GLP-1 receptor agonist (incretin mimetic)

GLP-1 S

GLP-1 Receptor Studies

GLP-1 S is a selective GLP-1 receptor agonist peptide. Its sequence is about 94 percent identical to the endogenous GLP-1 hormone, with one change that resists enzymatic cleavage. Research has measured insulin release, appetite signalling and gastric emptying. A fatty acid chain lets it bind albumin, which extends its half-life.

For laboratory research use only - not for human or animal use

Available in the Eon catalog - GLP-1 S from $85.00

Molecular data

Molecular formulaC187H291N45O59
Molecular weight4113.58 Da
SequenceHis-Aib-Glu-Gly-Thr-Phe-Thr-Ser-Asp-Val-Ser-Ser-Tyr-Leu-Glu-Gly-Gln-Ala-Ala-Lys(AEEA-AEEA-gGlu-C18 diacid)-Glu-Phe-Ile-Ala-Trp-Leu-Val-Arg-Gly-Arg-Gly
Sequence length31 residues
CAS / identifier910463-68-2
Physical formLyophilized powder
Available sizes20mg

How it works

GLP-1R

GLP-1 Receptor Agonism

Selectively binds GLP-1 receptors. Published characterisation describes glucose-dependent insulin secretion, glucagon suppression and delayed gastric emptying in study models. Insulin response scales with glucose, a property examined relative to non-incretin secretagogues.

  • Glucose-dependent insulin secretion
  • Glucagon suppression
  • Delayed gastric emptying
CNS

Central GLP-1R Signalling

Engages GLP-1 receptors in the hypothalamus and hindbrain, with hunger, satiety and energy intake as the measured endpoints.

  • Food intake measured
  • Satiety signalling measured
  • Lower caloric intake
PK

Extended Half-Life Design

A C18 fatty-diacid chain confers reversible albumin binding and resistance to DPP-4 degradation, extending the plasma half-life to roughly 7 days in research models.

  • ~165-hour half-life
  • Albumin-binding modification
  • DPP-4 resistant

What the research shows

Metabolic

Metabolic Receptor Research

GLP-1 receptor agonism is a principal focus of metabolic research, and GLP-1 S is a selective agonist used as a reference compound in that work.

Endocrine

Glycemic Pathway Research

GLP-1 S is studied for glucose-dependent insulin secretion and glycemic endpoints in metabolic research.

Cardiometabolic

Cardiovascular Outcomes

Cardiometabolic signalling is a further area of research interest for this receptor class, beyond glucose handling.

Neuroscience

Hypothalamic & Reward Circuitry

GLP-1 receptor signaling in the hypothalamus and hindbrain modulates satiety and food-reward pathways, a focus of ongoing neuroscience research.

Specification

Compound ClassGLP-1 receptor agonist (incretin mimetic)
Research NameGLP-1 S
TargetGLP-1 receptor (GLP-1R)
FormLyophilized powder
Molecular Weight4,113.58 g/mol
Purity≥99% (HPLC verified)
TestingThird-party HPLC, Mass Spec, Endotoxin
Half-Life~165 hours (~7 days)
Storage-20°C for long-term stability
SolubilityWater-soluble
COAIncluded with every order

Frequently asked questions

What is GLP-1 S?

GLP-1 S is a long-acting and selective GLP-1 receptor agonist. It mimics the incretin hormone GLP-1; published characterisation describes glucose-dependent insulin secretion, glucagon suppression, delayed gastric emptying and central appetite-pathway signalling.

How does it differ from GLP-2 TZ and GLP-3 RT?

GLP-1 S is a single-receptor (GLP-1) agonist. GLP-2 TZ is a dual GLP-1/GIP agonist, and GLP-3 RT is a triple GLP-1/GIP/glucagon agonist. The distinction is receptor coverage.

What is the molecular weight and purity?

GLP-1 S has a molecular weight of 4,113.58 g/mol. Every vial is supplied at ≥99% purity, verified by HPLC, with a Certificate of Analysis included.

How should it be stored?

Store lyophilized vials at -20°C for long-term stability, protected from light and moisture.

Is this product for human use?

No. GLP-1 S is sold strictly as a research compound for laboratory and in-vitro use only. It is not intended for human or animal consumption, diagnosis, or treatment.

For laboratory research use only. Not a drug, supplement, or medical product; not for human or animal use. All findings referenced are from published preclinical/laboratory research.